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ターゲット

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天然化合物

リコンビナントタンパク質

カタログ番号	製品名	別名	ターゲット
T22833	H-9 dihydrochloride		EGFR , 5-HT Receptor , PKA
	H-9 dihydrochloride is a potent protein kinase (PKA) inhibitor.H-9 Dihydrochloride significantly reduces the excitatory response to 5-HT at low concentrations.H-9 Dihydrochloride affects pharyngeal activity.H-9 Dihydroch...		EGFR , 5-HT Receptor , PKA
T21128	Lansoprazole sulfide	Lansoprazole impurity C,AG-1777,EC 600-451-9,H 225/18,K-1252
	Lansoprazole sulfide is an impurity of Lansoprazole, which is a gastric pump inhibitor.
T67324	(1'R,3a'R,8a'S,9'S,9a'S)-1'-Methyl-3'-oxo-N,N-diphenyl-3',3a',5',7',8',8a',9',9a'-octahydro-1'H-spiro[[1,3]dioxolane-2,6'-naphtho[2,3-c]furan]-9'-carboxamide
	(1'R,3a'R,8a'S,9'S,9a'S)-1'-Methyl-3'-oxo-N,N-diphenyl-3',3a',5',7',8',8a',9',9a'-octahydro-1'H-spiro[[1,3]dioxolane-2,6'-naphtho[2,3-c]furan]-9'-carboxamide is a useful organic compound for research related to life scie...
T7354	H-Val-Pro-Pro-OH		RAAS
	H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).		RAAS
T11526	DPP-IV-IN-2	H-Lys(4-nitro-Z)-pyrrolidide	DPP-4
	DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).		DPP-4
T33820	ORG 2766	ORG-2766,ORG2766
	ORG 2766 is an ACTH 4-9 (H-Met(O)-Glu-His-Phe-D-Lys-Phe-OH) analog and neurotrophic peptide.
T62297	H-Val-Pro-Pro-OH TFA
	H-Val-Pro-Pro-OH (TFA) is an inhibitor of angiotensin I converting enzyme (ACE) (IC50: 9 μM).H-Val-Pro-Pro-OH (TFA) is a milk-derived proline peptide derivative.
T25481	H 77	H77,H-77
	H 77 is a new effective renin inhibitor. H 77 is angiotensinogen (6-13)-octapeptide in which the peptide bond -CO-NH- at the Leu(9)-Leu(11) linkage is replaced by a -CH2-NH- bond.
T67578	H-Glu(OBzl)-OH
	H-Glu(OBzl)-OH is a useful organic compound for research related to life sciences. The catalog number is T67578 and the CAS number is 1676-73-9.
T63994	MMP-9-IN-4
	MMP-9-IN-4 is an inhibitor of MMP-9 and interacts with MMP-9 to form H-π with an IC50 value of 7.46 nM. MMP-9-IN-4 also inhibits AKT activity with an IC50 value of 8.82 nM. MMP-9-IN-4 induces apoptosis, shows cytotoxicit...
T67362	H-Glu(OtBu)-OH
	H-Glu(OtBu)-OH is a useful organic compound for research related to life sciences. The catalog number is T67362 and the CAS number is 2419-56-9.
TP1350	H-Val-Pro-Pro-OH TFA (58872-39-2 free base)	H-Val-Pro-Pro-OH TFA
	H-Val-Pro-Pro-OH(TFA), a proline peptide derivative from milk, is an ACE inhibitor with IC50 of 9 M.
T62156	HIV-1 integrase inhibitor 9
	HIV-1 integrase inhibitor 9 (compound 8a) is a potent inhibitor of HIV-1 RNase H (IC50: 12.3 μM) and has antiviral effects.
T67086	H-D-Thr(tBu)-OH
	H-D-Thr(tBu)-OH is a useful organic compound for research related to life sciences. The catalog number is T67086 and the CAS number is 201274-81-9.
T67312	H-DL-Phe(4-NO2)-OH
	H-DL-Phe(4-NO2)-OH is a useful organic compound for research related to life sciences. The catalog number is T67312 and the CAS number is 2922-40-9.
T66916	H-Cys(Acm)-OH HCl
	H-Cys(Acm)-OH HCl is a useful organic compound for research related to life sciences. The catalog number is T66916 and the CAS number is 28798-28-9.
T66595	H-Hyp-OMe hydrochloride
	H-Hyp-OMe hydrochloride is a useful organic compound for research related to life sciences. The catalog number is T66595 and the CAS number is 40216-83-9.
T65771	1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole
	1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole is a useful organic compound for research related to life sciences. The catalog number is T65771 and the CAS number is 152628-02-9.
T74621	STING agonist-9
	STING Agonist-9 (Compound 45) is a powerful stimulator of the STING pathway, demonstrating potent activity with an EC50 of 1.2 nM against human STING (h-STING) and 32.82 μM against mouse STING (m-STING). It exhibits anti...
T66626	H-D-Allo-Ile-OH
	H-D-Allo-Ile-OH is a useful organic compound for research related to life sciences. The catalog number is T66626 and the CAS number is 1509-35-9.
T65925	H-Asp(ome)-OMe HCl
	H-Asp(ome)-OMe HCl is a useful organic compound for research related to life sciences. The catalog number is T65925 and the CAS number is 32213-95-9.
T64955	H-DL-Phg(2-Cl)-OH
	H-DL-Phg(2-Cl)-OH is a useful organic compound for research related to life sciences. The catalog number is T64955 and the CAS number is 88744-36-9.
T64776	H-Phe(2,4-DiCl)-OH
	H-Phe(2,4-DiCl)-OH is a useful organic compound for research related to life sciences. The catalog number is T64776 and the CAS number is 111119-36-9.
T78388	9-Amino-6-chloro-2-methoxyacridine
	9-Amino-6-chloro-2-methoxyacridine serves as a pH-sensitive fluorescent probe commonly utilized to assess vacuolar pH variations upon substrate translocation across the tonoplast via a putative H+/solute antiport system ...
TP1727	Gp100 (25-33), human
	Gp100 (25-33), human is the amino acids 25-33 fragment of the human melanoma antigen. It is a 9-amino acid (AA) epitope restricted by H-2Db and recognized by the T cells.This is amino acids 25 to 33 fragment of human mel...
TP1416	Gp100 (25-33), human TFA (212370-40-6 free base)	Gp100 (25-33), human TFA
	Gp100 (25-33), human TFA is a 25-33 amino acid fragment of human melanoma antigen.Gp100 (25-33), human TFA is a 9-amino acid (AA) epitopes restricted by h-2db and recognized by T cells.
T78599	CK2-IN-9
	CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporter activity with an IC50 of 75 nM. In rats, it demonstrates low e...
T75766	GP(33-41) TFA
	GP(33-41) TFA, a 9-amino-acid (aa) peptide, represents the optimal sequence of the lymphocytic choriomeningitis virus GP1 epitope, effectively upregulating H-2D b molecules on the RMA-S (Db Kb) cell surface with a SC 50 ...
TP1752	GP(33-41)
	GP(33-41), a 9-aa-long peptide, is the optimal sequence of the GP1 epitope of lymphocytic choriomeningitis virus, and can upregulate H-2Db molecules at the RMA-S (Db Kb) cell surface with a SC50 of 344 nM. GP33-41 Epitop...
T37053	Z-(L-Arg)-AMC (hydrochloride)
	Z-(L-Arg)-AMC is a fluorogenic substrate for trypsin, cathepsin B, and cathepsin H.1,2Upon enzymatic cleavage by trypsin, cathepsin B, or cathepsin H, 7-amino-4-methylcoumarin (AMC) is released and its fluorescence can b...
T70988	Ibulocydine
	Ibulocydine is a potent CDK inhibitor. Ibulocydine has high activity against Cdk7/cyclin H/Mat1 and Cdk9/cyclin T. Ibulocydine inhibited the growth of HCC cells more effectively than other Cdk inhibitors, including olomo...
T36443	(R,R)-CXCR2-IN-2	(R,R)-CXCR2-IN-2
	(R,R)-CXCR2-IN-2, a diastereoisomer of CXCR2-IN-2 (compound 68), functions as a brain-penetrant CXCR2 antagonist. It exhibits a pIC50 of 9 in the Tango assay and 6.8 in the HWB Gro-α induced CD11b expression assay[1].
T36412	Multiflorenol
	Multiflorenol is a triterpene that has been found in T. kirilowii seeds.1 It inhibits in vitro activation of Epstein-Barr virus early antigen (EBV-EA) induced by the tumor promoter phorbol 12-myristate 13-acetate in a co...
T35549	Elsinochrome A
	Elsinochrome A is a perylenequinone fungal metabolite that has been found inHypomycesand has anticancer activity.1Photoactivation of elsinochrome A induces the production of singlet oxygen and apoptosis in R366.4 rhesus ...
T35451	β-Defensin-2 (human) (trifluoroacetate salt)
	β-Defensin-2 is a peptide with antimicrobial properties that protects the skin and mucosal membranes of the respiratory, genitourinary, and gastrointestinal tracts.1It inhibits the growth of periodontopathogenic and cari...
T35426	β-Defensin-1 (human) (trifluoroacetate salt)
	β-Defensin-1 is a peptide with antimicrobial properties that protects the skin and mucosal membranes of the respiratory, genitourinary, and gastrointestinal tracts.1It inhibits the growth ofB. adolescentis,L. acidophilus...
T35800	MD001
	MD001 is a dual agonist of peroxisome proliferator-activated receptor α (PPARα) and PPARγ.1 It binds to PPARα and PPARγ (Kds = 9.55 and 0.14 μM, respectively) but does not bind to PPARβ/δ at concentrations up to 500 μM. ...
T35504	(±)10-HDHA
	(±)10-HDHA is an autoxidation product of docosahexaenoic acid (DHA) in vitro.[1][2] It is also produced from incubations of DHA in rat liver, brain, and intestinal microsomes.[3][4][5] (±)10-HDHA is a potential marker of...
T37847	Zonisamide-13C2,15N	Zonisamide-13C2,15N
	Zonisamide-13C2,15N is intended for use as an internal standard for the quantification of zonisamide by GC- or LC-MS. Zonisamide is an antiepileptic agent.1 It selectively inhibits the repeated firing of sodium channels ...
T35799	MBX-8025 (sodium salt)
	MBX-8025 is an agonist of peroxisome proliferator-activated receptor δ (PPARδ).1 It is greater than 750- and 2,500-fold selective for PPARδ over PPARα and PPARγ. MBX-8025 (10 mg/kg per day for eight weeks) reduces increa...
T38042	Resolvin D4	Resolvin D4,RvD4
	Resolvin D4 (RvD4) is a specialized pro-resolving mediator derived from docosahexaenoic acid . [1] It has been detected in human milk, in the dorsal pouch of mice before and after infection with S. aureus, and in untreat...
T38145	Eltoprazine
	Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.IC50 value:Target: 5-HT1A/1B agonist; 5-HT2C antagonistin vitro...
T37741	N-hexadecanoyl-L-Homoserine lactone	C16-HSL,N-palmitoyl-L-Homoserine,N-hexadecanoyl-L-Homoserine lactone
	Quorum sensing is a regulatory system used by bacteria for controlling gene expression in response to increasing cell density.[1] This regulatory process manifests itself with a variety of phenotypes including biofilm fo...
T36570	KUS121
	KUS121 is a valosin-containing protein (VCP) modulator that inhibits VCP ATPase activity (IC50= 330 nM).1It inhibits cell death, ATP depletion, and upregulation of C/EBP-homologous protein (CHOP) induced by tunicamycin, ...

Compounds

H-9 dihydrochloride

T22833

Synonym:

Target: EGFR, 5-HT Receptor, PKA

Lansoprazole sulfide

T21128

Synonym: Lansoprazole impurity C,AG-1777,EC 600-451-9,H 225/18,K-1252

Target:

(1'R,3a'R,8a'S,9'S,9a'S)-1'-Methyl-3'-oxo-N,N-diphenyl-3',3a',5',7',8',8a',9',9a'-octahydro-1'H-spiro[[1,3]dioxolane-2,6'-naphtho[2,3-c]furan]-9'-carboxamide

Synonym: H-Lys(4-nitro-Z)-pyrrolidide

Target: DPP-4

ORG 2766

T33820

Synonym: ORG-2766,ORG2766

H-Val-Pro-Pro-OH TFA (58872-39-2 free base)

TP1350

Synonym: H-Val-Pro-Pro-OH TFA

Target:

HIV-1 integrase inhibitor 9

H-Hyp-OMe hydrochloride

T66595

Synonym:

Target:

1,7'-Dimethyl-2'-propyl-1H,1'H-2,5'-bibenzo[d]imidazole

9-Amino-6-chloro-2-methoxyacridine

Gp100 (25-33), human TFA (212370-40-6 free base)

TP1416

Synonym: Gp100 (25-33), human TFA

Z-(L-Arg)-AMC (hydrochloride)

Synonym: (R,R)-CXCR2-IN-2

β-Defensin-2 (human) (trifluoroacetate salt)

T35451

Synonym:

Target:

β-Defensin-1 (human) (trifluoroacetate salt)

Synonym: Zonisamide-13C2,15N

Target:

MBX-8025 (sodium salt)

Synonym: Resolvin D4,RvD4

N-hexadecanoyl-L-Homoserine lactone

T37741

Synonym: C16-HSL,N-palmitoyl-L-Homoserine,N-hexadecanoyl-L-Homoserine lactone

カタログ番号	製品名	ターゲット
T3S1641	Esculentoside H	TNF , NF-κB , JNK
	Phytolaccaceae has anti-tumor activity, the mechanism may be related to the capacity of Esculentoside H for TNF release.	TNF , NF-κB , JNK
T36914	2-Hydroxyanthraquinone	Others
	2-Hydroxyanthraquinone is an anthraquinone that has been found inSpermacoce latifoliaand has antibacterial and estrogenic activities.1,2It is active againstB. subtilisandB. cereus(MICs = 1.9 and 62.5 μg/ml, respectively)...	Others
TN4378	Kanshone H	Others
	Kanshone H is a natural product for research related to life sciences. The catalog number is TN4378 and the CAS number is 1445952-33-9.	Others
TN3318	9-Hydroxy-alpha-lapachone	Antifection
	9-Hydroxy-alpha-lapachone can highly inhibit the growth of H. pylori, it exhibits potent inhibitory activity against H. pylori Cystathionine gamma-synthase, with IC(50) values of 4.64 microM. It may have anti-inflammator...	Antifection
T36438	Sporogen-AO 1
	Sporogen-AO 1 is a fungal metabolite originally isolated fromA. oryzaethat has diverse biological activities.1,2,3,4,5It inhibits HIV-1 Tat transactivation in a cell-based assay with an IC50value of 15.8 μM.4Sporogen-AO ...
T36348	Cerebroside C
	Cerebroside C is a fungal metabolite and glycosphingolipid that has been found in the rice pathogenic fungusM. grisea.1It induces production of the phytoalexin momilactone A when applied to wounded rice leaves, indicatin...

天然物製品

Esculentoside H

T3S1641

Synonym:

Target: TNF, NF-κB, JNK

2-Hydroxyanthraquinone

9-Hydroxy-alpha-lapachone

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-03274	CXCL11 Protein, Human, Recombinant	Human	E. coli
	I-TAC, also known as CXCL11, is a small cytokine belonging to the CXC chemokine family. It is highly expressed in peripheral blood leukocytes, pancreas and liver, with moderate levels in thymus, spleen and lung and low e...
TMPY-06872	Ara h 9 Protein, Arachis hypogaea, Recombinant	Arachis hypogaea	P. pastoris (Yeast)
	Ara h 9 Protein, Arachis hypogaea, Recombinant is expressed in P. pastoris yeast expression system. The predicted molecular weight is 16.34 kDa.
TMPY-04989	Galectin-9 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	LGALS9 (Galectin 9) is a Protein Coding gene. 6 alternatively spliced human isoforms have been reported. The galectins are a family of beta-galactoside-binding proteins implicated in modulating cell-cell and cell-matrix ...
TMPJ-00865	VEGF121 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Human VEGF121, also known as Vascular endothelial growth factor A, VEGFA, Vascular permeability factor, VPF and VEGF, is a homodimeric, heparin-binding glycoprotein which belongs to the platelet-derived growth factor (PD...
TMPY-03698	VEGF121b Protein, Human, Recombinant	Human	HEK293 Cells
	VEGF121b Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 34.10 kDa and the accession number is P15692-9.
TMPH-00005	YAP1 Protein, Human, Recombinant (Isoform 9, His)	Human	P. pastoris (Yeast)
	YAP1 Protein, Human, Recombinant (Isoform 9, His) is expressed in yeast with C-6xHis tag. The predicted molecular weight is 56.4 kDa; 80 kDa, reducing conditions and the accession number is P46937-9.
TMPY-00818	Granzyme H/GZMH Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Granzymes are key components of the immune response that play important roles in eliminating host cells infected by intracellular pathogens. Several granzymes are potent inducers of cell death. A total of eight granzymes...
TMPJ-01306	CFHR5 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Complement factor H-related protein 5(FHR-5 for short), is a secreted protein which contains 9 Sushi (CCP/SCR) domains. It is expressed by the liver and secreted in plasma. The pattern of the deposits is similar to other...
TMPK-00825	VEGF121 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	Vascular endothelial growth factor (VEGF or VEGF-A), also known as vascular permeability factor (VPF), is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. VEGF165 appears to be the most a...
TMPK-00826	VEGF121 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	Vascular endothelial growth factor (VEGF or VEGF-A), also known as vascular permeability factor (VPF), is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. VEGF165 appears to be the most a...
TMPY-05268	Neurofascin Protein, Human, Recombinant (hFc), Biotinylated	Human	HEK293 Cells
	Neurofascin Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 130 kDa and the accession number is O94856-9.
TMPK-01413	H-2K (b) &B2M&OVA (SIINFEKL) Monomer Protein, Mouse, MHC (His & Avi)	Mouse	HEK293 Cells
	Ovalbumin (OVA) has been historically a popular source of such antigens, since OVA can induce both humoral and cellular immune responses based on well-characterised peptide epitopes. The OVA257-264 octapeptide was one of...
TMPK-01535	Chimeric HLA-A*02:01 (mα3) &B2M&LMP2 (CLGGLLTMV) Tetramer Protein, Human&Mouse, MHC (His & Avi)	Human & Mouse	HEK293 Cells
	The immunoproteasome, having been linked to neurodegenerative diseases and hematological cancers, has been shown to play an important role in MHC class I antigen presentation. The development of molecular probes that sel...
TMPK-01534	Chimeric HLA-A*02:01 (mα3) &B2M&LMP2 (CLGGLLTMV) Monomer Protein, Human&Mouse, MHC (His & Avi)	Human & Mouse	HEK293 Cells
	The immunoproteasome, having been linked to neurodegenerative diseases and hematological cancers, has been shown to play an important role in MHC class I antigen presentation. The development of molecular probes that sel...
TMPK-01522	Chimeric HLA-A*02:01 (mα3) &B2M&WT-1 (RMFPNAPYL) Tetramer Protein, Human&Mouse, MHC (His & Avi)	Human & Mouse	HEK293 Cells
	The WT1 protein plays a role in cell growth, the process by which cells mature to perform specific functions (differentiation), and the self-destruction of cells (apoptosis). WT1 is differentially expressed in serous, en...
TMPK-01523	Chimeric HLA-A*02:01 (mα3) &B2M&WT-1 (RMFPNAPYL) Monomer Protein, Human&Mouse, MHC (His & Avi)	Human & Mouse	HEK293 Cells
	The WT1 protein plays a role in cell growth, the process by which cells mature to perform specific functions (differentiation), and the self-destruction of cells (apoptosis). WT1 is differentially expressed in serous, en...